Overview and History Methyltestosterone

Methyltestosterone is unquestionably a typical anabolic steroid. It's classic not just in terms of the outcomes and impacts it can bring individuals in terms of mass building and performance capabilities, but it's also a true old-school compound. While many individuals may not refer to it by its full name, the reality is that most people are aware of it without even realizing it.

It is a steroid that truly works, and it is quite powerful and efficient in terms of its effects on the human body. It is not only one of the oldest steroids in history, but it is also one of the most important steroids in history. This is due to the fact that it was the first synthetic form of testosterone.

This is present in certain synthetic versions, but it was the first true, raw form of testosterone, the androgenic hormone generated endogenously within the male body. The earliest version of this steroid was simply the hormone without an ester attached, which was very similar to Testosterone Suspension, sometimes known as Test Susp in bodybuilding circles. Testosterone Propionate, sometimes known as Test Prop, would become life and enter the open market with its kin in 1937.

Although Ciba's Metandren was a profitable medicine, the most well-known brand is no longer accessible. Currently, generic brands, as well as many underground lab formulations, are the most common. For numerous years, Teston has been the only name brand pharmaceutical-based pure Methyltestosterone available.

While methyltestosterone is not as widespread on the pharmaceutical market as it once was, it is nevertheless utilized in some parts of the world. Despite the fact that it has been removed from several markets and that many US physicians seldom prescribe it, methyltestosterone is an insignificant supply in the US pharmaceutical market. The chemical has been used to treat low testosterone, andropause, and cryptorchidism in males.

It has also been used to manage excess lactation after pregnancy and osteoporosis in some breast cancer treatment schemes. Most notably, Methyltestosterone has shown some effectiveness in treating menopause by restoring frequently lost libido and energy levels, which often decline during this time of life for many women. While methyltestosterone has been successful in menopausal therapy in the modern period, most women are now taking different types of testosterone. The most prevalent are creams and gels. Testosterone and progesterone creams, as well as subcutaneous implant pellets like Testopel, have proved extremely effective.

While it has had some success, Methyltestosterone is one of the most contentious testosterone medicines in conventional medicine. The main source of contention is its hepatotoxicity, which is not shared by other testosterone derivatives.

Furthermore, unlike other testosterone compounds, Methyltestosterone is rarely utilized in performance-boosting circles. Methyltestosterone, like other testosterone molecules, has an estrogenic character, but it is much more apparent in this form, making it a bad choice for most sportsmen.

Chemistry Behind Methyltestosterone

  • [17alpha-methyl-4-androstene-3-one,17b-ol]
  • Molecular Weight: 302.4558
  • Formula: C20H30O2
  • Melting Point: 162-167
  • Manufacturer: Most Major Pharmaceutical Companies
  • Effective dose: (Men) 25-100mgs/day; (Women) N/A
  • Active Life: 6-8 hours
  • Detection Time: 4-6 weeks
  • Anabolic /Androgenic Ratio (Range): 94-130/115-150
Chemical Structure of Methyltestosterone


Methyltestosterone is the first oral testosterone preparation and the first C17-alpha-alkylated (C17-aa) steroid ever created. The compound has appeared under a variety of trade names throughout the years, but Ciba's Metandren is possibly the most well-known Methyltestosterone compound of all time.

Ciba's Methyltestosterone, while oral, was a sublingual version, which increased the testosterone hormone's absorption. In fact, as compared to a pill version, this form doubles bioavailability and allows the individual to attain peak testosterone levels in an hour. When Methyltestosterone is taken as a pill, peak levels can take up to two hours to achieve, not to mention the substantially decreased potency.

Methyltestosterone is a pure derivative of the hormone testosterone, but what distinguishes it is the addition of a methyl grouping on top to guarantee it can be taken in and absorbed orally.

The methyl group added to the molecule guarantees that the testosterone survives digestion and mechanical breakdown inside the body. If we only consider it as a testosterone hormone, Methyltest is excellent since it is a synthetic replica of the original male androgen that we all know and adore. 

The fact is that the body cannot distinguish the difference, and it will attach to androgen receptors as if it were your body's own endogenously generated testosterone.

Because Methyltestosterone is testosterone in its purest form, it will perform just as well as the original testosterone formulation. Apart from the obvious physical needs, it is critical to supplement with testosterone for cognitive or cerebral reasons.

While Methyltestosterone is important to understand, it's also a good idea to examine alternative test profiles such as Testosterone Cypionate, Testosterone Enanthate, Testosterone Propionate, or even the aforementioned test suspension.

Effects of Methyltestosterone

Exogenous administration of Methyltestosterone causes its effects by simply raising the number of circulating androgens. This might be done to battle a condition caused by low levels, or it could be done to raise androgen levels above baseline levels to aid in the treatment of another ailment.

While both are conceivable in a medical context, the former is more typical. By supplementing with this androgen, the benefits of Methyltestosterone should improve the individual's sex drive and energy levels, which are generally reduced when the hormone is low in the body. We will, however, discover that the steroid is not nearly as harmful as many had incorrectly assumed, but it will still be unsuitable for long-term performance usage.

The benefits of Methyltestosterone will largely help athletes from an androgenic, rather than anabolic, perspective. The high amount of androgenic activity might considerably enhance hostility by supplementing for brief periods of time with a big dose. This might help powerlifters and other strength athletes prepare for competition.

However, there is something we need to clarify when looking at the effects of Methyltestosterone in this area. It's also worth noting that aggressiveness isn't always a bad thing. What we do with hostility determines whether it is right or bad.

When employed appropriately, such as in strength competitions, increased hostility may be tremendously advantageous. Some bodybuilders may find the benefits of Methyltestosterone advantageous in this regard shortly before a competition to assist them to get through the final phases when energy levels are frequently low. However, because of Methyltestosterone's strong estrogenic action, there are usually better alternatives.

Side Effects Methyltestosterone

For most adult males, the testosterone hormone is a fairly side effect friendly hormone. However, the negative effects of Methyltestosterone might be higher and harsher than those of other testosterone derivatives. This is true for most regions that may be negatively affected by testosterone. To assist you to understand the potential side effects of Methyltestosterone, we've divided them into categories and provided all of the information you'll need.

Estrogenic: Methyltestosterone's potential adverse effects include estrogenic effects. These effects are caused by testosterone converting to oestrogen because of its interaction with the aromatase enzyme.  Because of the 17-alpha methylation of the hormone, methyltestosterone aromatizes slower than other testosterone molecules, but instead of converting to estradiol, it converts to methyl estradiol.

Methylestradiol is a very potent estrogenic hormone, which can cause gynecomastia and water retention. All testosterone hormones can cause these consequences, but Methyltestosterone has a larger chance of doing so.

Indeed, the estrogenic side effects of Methyltestosterone can arise apparently overnight, necessitating the usage of an anti-estrogen when males use this testosterone.

Selective Estrogen Receptor Modulators or Aromatase Inhibitors are two possibilities for addressing the estrogenic side effects of Methyltestosterone. SERMs, such as Tamoxifen Citrate, work by binding to oestrogen receptors, inhibiting the oestrogen hormone from binding and activating. 

AIs, such as Letrozole, work by blocking the aromatase mechanism, lowering blood oestrogen levels. AIs are by far the most effective, although they can have an adverse effect on cholesterol. As a result, some people may benefit from using a 5-alpha reductase inhibitor like Finasteride. A 5-alpha reductase inhibitor will lower the androgenicity of the hormone; it will not be fully eliminated, but it will be significantly reduced.

Women must likewise be concerned about Methyltestosterone's androgenic adverse effects. This steroid has a high virilization potential, which might manifest as body hair growth, voice chord deepening, and clitoral enlargement. Low dosages of the hormone combined with esterified estrogens can lower the likelihood of virilization, such as the product Estratest, which has a very low amount of Methyltestosterone as well as the essential esterified oestrogen. Most women, however, are advised to quit usage promptly if virilization signs appear.

If the medication is stopped as soon as the symptoms appear, they will go away quickly. Ignoring the signs may result in irreparable damage. Because of the steroid's high virilization potential, no woman should use Methyltestosterone for performance goals. This steroid should be used in extremely low dosages only in certain therapeutic situations.

Cardiovascular: High blood pressure is one of the adverse effects of Methyltestosterone, however, it is generally reduced when the user reduces water retention. High amounts of water retention are renowned for increasing hypertension. Most people will not have a problem if their water retention is addressed; nevertheless, high blood pressure is still possible but improbable.

Methyltestosterone, like other testosterone molecules, has a detrimental effect on cholesterol. Most testosterone hormones have a little effect on HDL cholesterol, giving mild suppression. As a cholesterol antioxidant supplement, it is recommended to take fish oil on a daily basis.

Testosterone: The majority of anabolic androgenic drugs inhibit natural testosterone synthesis. The rate of suppression, however, is dependent on the steroid in issue and can also be influenced by the total dosage. While Methyltestosterone is considerably suppressive, the individual should be able to prevent low testosterone since Methyltestosterone will provide all the testosterone he requires. He will, however, be in a low state after usage is ended.

Most men are urged to pursue a Post Cycle Therapy regimen once all use has been ceased. This will increase natural production and lower the likelihood of a low testosterone condition significantly. Those who are healthy can recover without a PCT plan, but it will take much longer and can be harmful to their health if a low level is maintained for an extended period of time.

Except for two instances, there is no need to forego a PCT strategy. Women will not be required to follow a PCT plan. Men suffering from low testosterone will also not require a PCT regimen, since such a condition would necessitate ongoing and indefinite testosterone medication to keep the problem at bay.

Hepatotoxicity: Methyltestosterone is hepatotoxic, although not in the way that many people believe. All C17-aa steroids are toxic to the liver, however, the degree of toxicity varies from steroid to steroid.

Therapeutic level dosages will cause some stress on the liver, and liver enzyme readings will rise with usage, but if the liver was healthy, to begin with, no harm should be done.

Cycles And Usage of Methyltestosterone

Methyltestosterone is quite powerful when dosed. If you want to boost your aggressiveness and athletic performance, stick to a 40-50 mg dose for no more than 8 weeks.

In a therapeutic environment, 10-40 mg is sufficient to reap the majority of the advantages. Most of the time, the initial doses will be greater, and they will gradually decrease until they reach the 10mg level.

Doses of methyltestosterone for females should be extremely low. No more than 2.5 mg, and even that may be too much for some ladies. Women who are prescribed or choose to use methyl tests are frequently given oestrogen pills to stack with the testosterone alone.

How To Buy Methyltestosterone

It is often encountered in the pharmaceutical industry because of its popularity in therapeutic settings. It's quite hard to get it on the black market or through UGLs but be warned: a lot of imitation steroids offered as Anadrol, Dianabol, or Winstrol are really simply Methyltestosterone, but if you know your steroids, you'll be able to detect an imposter batch of Methyltest from a mile away.

Methyltestosterone Purchase Online

You will need a doctor's prescription to obtain it. However, if you try to acquire it, you will find that it is rarely sold by UGLs or black-market dealers. Remember that purchasing steroids is unlawful under the Controlled Substances Act and the Steroid Act of 1990, as amended in the early 2000s.

Methyltestosterone can be easily obtained online. While most big internet providers do not carry it, there are some that do, and if you really want it, you can locate it. Furthermore, because it is manufactured by a multitude of reputable pharmaceutical businesses, there should be no need to ever buy an illegal version.

While it is possible to purchase Methyltestosterone online, we do not advocate it. The Steroid Control Act of 1990 categorised anabolic androgenic steroids as Schedule III restricted drugs in the United States. The Steroid Control Act of 2004 would subsequently strengthen this regulation, and individuals who violate it would face significant penalties and prison time.

Outside of the United States, some countries are similarly rigorous, while many are considerably more liberal. Many nations allow anabolic steroids to be purchased over the counter without a prescription, although most do not allow internet purchases. If you want to buy anabolic steroids legally, you must get them through a pharmacy. While legality is frequently significantly more permissive in many nations, there can be exceptions and variations based on the country in question. As a result, it is critical that you completely grasp the laws of the nation in which you live before making any anabolic steroid purchases. 

Review on Methyltestosterone

Methyltestosterone is a one-of-a-kind testosterone molecule on the market. In reality, whereas different testosterone molecules all have a somewhat different nature, most are almost identical outside of Methyltestosterone.

Methyltestosterone is distinct due to its lack of anabolic power, increased translatable androgenicity, and estrogenic properties. When we examine its C17-aa character, it actually distinguishes itself from the majority of testosterone molecules.

While methyltestosterone is unusual in origin, it is likewise unusual in its application. While there is a performance objective for some, when we analyse efficacy, we will find that there are far superior solutions. While useful as therapeutic testosterone for a male patient, it is frequently reported to be weak in comparison to most testosterone compounds.

Most men will be happier with injectable testosterone, testosterone gels, and, in some circumstances, testosterone implant pellets. The sole genuine advantage of this hormone molecule appears to be in female usage to counteract the symptoms of menopause, but only when combined with esterified oestrogen at modest dosages. It appears to have a lot of potential in this application and might become a regular element of many female hormone replacement therapy schemes. However, in the present era, it is far from the only alternative, and as this field of medicine develops, it may become obsolete in the near future.

  • Ziller33 Avatar
    Ziller3318 days ago

    Thanks for the info

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